Important (for sprays)! Before screwing on the dispenser, remove the protective ring from the bottle cap.
Relax Support
Soft modulation of NMDA receptors without side philosophizing.
Spray, 10 ml
100 mcg Glyx-13 per press
55 doses in one bottle
What's inside:
Glyx-13 (rapastinel), 100 mcg/press
A peptide that communicates with the NMDA receptor like a smart introvert: activates - but does not cross the line.
Works not as an antagonist, but as a “psychotherapist with access to the glycine site”.
Capable of increasing neuroplasticity without sedation, hallucinations and the desire to go to Peru for ayahuasca.
Biochemistry of action:
1. Glyx-13 binds to the glycine co-agonist site of the NMDA receptor
→ does not fully activate it, but optimizes the opening of the ion channel.
2. This causes a moderate and safe entry of Ca²⁺ into the postsynaptic neuron
→ stimulation of CREB and expression of neurotrophins, especially BDNF.
3. The neuroplasticity cascade is triggered (mTOR, MAPK, CaMKII),
→ synaptic transmission is improved, especially in the prefrontal cortex and hippocampus.
4. Simultaneously inhibits NMDA overactivity associated with anxiety and neuroinflammation
→ without “overkill” and psychodissociation (unlike ketamine or memantine).
Form and dosage:
spray (tasteless, like most small existential solutions)
1-2 presses in the evening or "on alarm"
Clinical effects:
Reduction of anxiety, panic expectations, neurovegetative tension
Improvement of adaptation to stress, emotional regulation
Support for neuroplasticity in depression and post-stress disorders
Increase in cognitive flexibility, decrease in rigidity of thinking
Without addiction, without sedation, without the effect of "inhibition"
Why is it needed:
When the anxious dominant does not turn off even in sleep
When serotonin has already tried, and GABA just ran away
When "everything is fine" - but only according to tests
Slogan:
Relax Support - calming worthy of your synapse.